United States
LY2183240 CAS NO.874902-19-9
- FOB Price: USD: 50.00-50.00 /Kilogram Get Latest Price
- Min.Order: 10 Gram
- Payment Terms: T/T,Other
- Available Specifications:
5(5-1000)Kilogram
- Product Details
Keywords
- LY2183240
- 874902-19-9
Quick Details
- ProName: LY2183240
- CasNo: 874902-19-9
- Appearance: white
- Application: Not for Human consumption
- DeliveryTime: 3 days
- PackAge: aluminium foil paper
- Port: Nanjing
- ProductionCapacity: 5000 Kilogram/Month
- Purity: 99.8%
- Storage: Safe
- Transportation: AIr
- LimitNum: 10 Gram
Superiority
LY2183240 is a potent, competitive inhibitor of anandamide uptake (IC50 = 270 pM; Ki = 540 pM) and hydrolysis.It increases anandamide levels in rat cerebellum (ED50 = 1.37 mg/kg) and displays dose-dependent efficacy (3-30 mg/kg) in several rodent models of persistent pain.
Details
LY-2183240 is a chemicals which acts both as a potent inhibitor of the reuptake of the endocannabinoid anandamide and as an inhibitor of fatty acid amide hydrolase, the primary enzyme responsible for degrading anandamide.